可逆性抑制剂

  • 网络reversible inhibitor;irreversible inhibitor;RIMA
可逆性抑制剂可逆性抑制剂
  1. 盐酸多奈哌齐是近年来应用于临床的一种新型可逆性胆碱酯酶抑制剂,用于治疗轻中度AD,国内外报道其具有一定疗效。

    Donepezil is a new reversible acetylcholinesterase inhibitor which is used to treat mild-moderate AD in clinical trials recent years .

  2. 该类具有代表性的杀虫剂主要有机磷农药和氨基甲酸酯类农药,而这些非可逆性的抑制剂对环境和人类都有很大的危害。

    The representative pesticides are organophosphorus and carbamate derivates , however , this kind of pesticide are harmful for the environment and human beings .

  3. 结论加可逆性激活抑制剂后,冻干前预处理血小板过程对血小板的功能活性没有显著影响。

    Conclusion The preprocessing before platelets lyophilization has no significant effects on the function and activity of platelets when the platelets activation inhibitor is added .

  4. 经过系统药理学研究表明,该生物碱具有良好抗胆碱酯酶效应,从而可认为该生物碱系一种新结构类型的可逆性胆碱酯酶抑制剂。

    The systematic pharmacological study shows that this alkaloid possesses good anticholinesterase effect , and therefore it is a new structure type of reversible acetylcholinesterase inhibitor .

  5. 56例仅接受放疗或同时服用抗胆碱酯酶剂,可以作为组内自身对照,证实放疗疗效较好。可逆性胆碱酯酶抑制剂的研究:2-氧化-1,3,2-二氧磷杂环己烷类化合物的合成

    56 cases were treated only by radiation or by combination of radiation and anticholinesterase drugs as self control in this group . STUDY ON REVERSIBLE ANTICHOLINESTERASE AGENTS : SYNTHESIS OF DERIVATIVES OF 1 , 3 , 2-DIOXAPHOSPHORINANE 2-OXIDE